SE9301732D0 - NEW CENTRALLY ACTING 5-, 6-, 7-, AND 8-SUBSTITUTED SULPHONE ESTERS OF N-MONOSUBSTITUTED 2-AMINOTETRALINS - Google Patents

NEW CENTRALLY ACTING 5-, 6-, 7-, AND 8-SUBSTITUTED SULPHONE ESTERS OF N-MONOSUBSTITUTED 2-AMINOTETRALINS

Info

Publication number
SE9301732D0
SE9301732D0 SE9301732A SE9301732A SE9301732D0 SE 9301732 D0 SE9301732 D0 SE 9301732D0 SE 9301732 A SE9301732 A SE 9301732A SE 9301732 A SE9301732 A SE 9301732A SE 9301732 D0 SE9301732 D0 SE 9301732D0
Authority
SE
Sweden
Prior art keywords
aminotetralins
monosubstituted
esters
centrally acting
new centrally
Prior art date
Application number
SE9301732A
Other languages
Swedish (sv)
Inventor
Vilhelm *Wikstroem Haakan
Original Assignee
Haakan Wilhelm Wikstroem
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Haakan Wilhelm Wikstroem filed Critical Haakan Wilhelm Wikstroem
Priority to SE9301732A priority Critical patent/SE9301732D0/en
Publication of SE9301732D0 publication Critical patent/SE9301732D0/en
Priority to AU68110/94A priority patent/AU6811094A/en
Priority to PCT/SE1994/000465 priority patent/WO1994026703A1/en

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

A compound of formula (1) or pharmaceutically acceptable acid addition salts thereof, wherein R1 is H, (C1-C8) alkyl, alkenyl, alkynyl, cyclopropylalkyl or (C1-C8) haloalkyl; X is CH2, O or S; R2-SO2-O is in position 5, 6, 7 or 8 and R2 is CF3, CF2CF3, C1-C8 alkyl, substituted aryl (e.g. 4-toluyl); R3 is H, CH3 or CH2CH3. When R3 is CH3 or CH2CH3, it is always in a cis-relationship with respect to the 2-amine substituent.
SE9301732A 1993-05-18 1993-05-18 NEW CENTRALLY ACTING 5-, 6-, 7-, AND 8-SUBSTITUTED SULPHONE ESTERS OF N-MONOSUBSTITUTED 2-AMINOTETRALINS SE9301732D0 (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
SE9301732A SE9301732D0 (en) 1993-05-18 1993-05-18 NEW CENTRALLY ACTING 5-, 6-, 7-, AND 8-SUBSTITUTED SULPHONE ESTERS OF N-MONOSUBSTITUTED 2-AMINOTETRALINS
AU68110/94A AU6811094A (en) 1993-05-18 1994-05-18 New centrally acting 5-, 6-, 7-, and 8-substituted sulphone esters of n-monosubstituted 2-aminotetralins and related structures
PCT/SE1994/000465 WO1994026703A1 (en) 1993-05-18 1994-05-18 New centrally acting 5-, 6-, 7-, and 8-substituted sulphone esters of n-monosubstituted 2-aminotetralins and related structures

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9301732A SE9301732D0 (en) 1993-05-18 1993-05-18 NEW CENTRALLY ACTING 5-, 6-, 7-, AND 8-SUBSTITUTED SULPHONE ESTERS OF N-MONOSUBSTITUTED 2-AMINOTETRALINS

Publications (1)

Publication Number Publication Date
SE9301732D0 true SE9301732D0 (en) 1993-05-18

Family

ID=20390003

Family Applications (1)

Application Number Title Priority Date Filing Date
SE9301732A SE9301732D0 (en) 1993-05-18 1993-05-18 NEW CENTRALLY ACTING 5-, 6-, 7-, AND 8-SUBSTITUTED SULPHONE ESTERS OF N-MONOSUBSTITUTED 2-AMINOTETRALINS

Country Status (3)

Country Link
AU (1) AU6811094A (en)
SE (1) SE9301732D0 (en)
WO (1) WO1994026703A1 (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9601110D0 (en) * 1996-03-22 1996-03-22 Astra Ab Substituted 1,2,3,4-tetrahydronaphthalene derivatives
DE10334188B4 (en) 2003-07-26 2007-07-05 Schwarz Pharma Ag Use of rotigotine to treat depression
DE10359528A1 (en) 2003-12-18 2005-07-28 Schwarz Pharma Ag (S) -2-N-propylamino-5-hydroxytetralin as a D3 agonist therapeutic
DE10361258A1 (en) 2003-12-24 2005-07-28 Schwarz Pharma Ag Use of substituted 2-aminotetralins for the preventive treatment of Parkinson's disease
DE102004014841B4 (en) 2004-03-24 2006-07-06 Schwarz Pharma Ag Use of rotigotine for the treatment and prevention of Parkinson-Plus syndrome
GB0426061D0 (en) * 2004-11-26 2004-12-29 Pfizer Ltd Chroman compounds
CA2703561C (en) 2007-11-28 2016-01-19 Ucb Pharma Gmbh Novel polymorphic form of rotigotine and process for production
IT1392387B1 (en) * 2008-09-26 2012-03-02 Solmag S P A Ora Fidia Farmaceutici S P A PROCESS FOR ROTIGOTINE PREPARATION

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE8605504D0 (en) * 1986-12-19 1986-12-19 Astra Laekemedel Ab NOVEL CHROMAN DERIVATIVES
ZA901277B (en) * 1989-02-27 1991-10-30 Lilly Co Eli Ring-substituted 2-amino-1,2,3,4-tetrahydronaphthalenes and 3-aminochromanes
SE8901889D0 (en) * 1989-05-26 1989-05-26 Astra Ab NOVEL 8-SUBSTITUTED-2-AMINOTETRALINES
SE8904361D0 (en) * 1989-12-22 1989-12-22 Astra Ab NEW CHROMAN AND THIOCHROMAN DERIVATIVES
KR100207876B1 (en) * 1990-10-12 1999-07-15 로버트 에이. 아미테이지 Therapeutically useful 2-aminotetralin derivatives

Also Published As

Publication number Publication date
WO1994026703A1 (en) 1994-11-24
AU6811094A (en) 1994-12-12

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